Contents

Russian Journal of Bioorganic Chemistry

Vol. 49, No. 1, 2023

5-Alkyloxymethyl Derivatives of 2ʹ-Deoxyuridine Bearing 2,4-Dinitrophenyl and Dansyl Groups: Synthesis and Antibacterial Activity

D. A. Makarov, I. A. Oskolsky, M. V. Jasko, P. N. Solyev, B. F. Vasilyeva, M. V. Demiankova, O. V. Efremenkova, S. N. Kochetkov, and L. A. Alexandrova p. S1  abstract

Innovative Technology of the Self-Emulsifying Drug Delivery System of the Anticonvulsant Galodif

V. U. Kuksenok, V. V. Shtrykova, V. D. Filimonov, T. V. Shushpanova, N. A. Bokhan, L. Seilerová, B. Kratohvil, and V. Sieberová p. S8  abstract

Triazole Moieties as Potent Drug Molecules: Synthetic Approaches and Application as Promising Candidates as Anticancer Agents (A Review)

V. K. Vashistha, A. Mittal, R. Bala, and R. V. S. R. Pullabhotla p. S13  abstract

A Brief Review on Schiff Base, Synthesis, and Their Antimicrobial Activities

Ruaa M. Dhedan, Sanaa A. Alsahib, and Rana Abid Ali p. S31  abstract

Virtual Screening of Orally Active Lead Compounds of Pearl Millet and Their Structural Activity Against Target Protein of COVID-19

Adarsh Kumar Shukla, and Ashwani Kumar p. S53  abstract

Synthesis and Biological Evaluation of Fused [1,2,3]Triazolo[4ʹ,5ʹ:4,5]pyrido[2,3-d]pyrimidine Linked 1,2,3-Triazolesas Potent EGFR Targeting Anticancer Agents

Sandhya Rani Bandi, T. Madhukar Reddy, Uma Rani Janapatla, and Sirassu Narsimha p. S71  abstract

Exploration of 2-(Substituted Phenyl)-thiazolidin-4-one as Anticancer Agents

Rahul B. Shinde, Dattatraya N. Pansare, Aniket P. Sarkate, Shailee V. Tiwari, Rohini N. Shelke, Deepak Lokwani, Shirish Jain, and Ashok M. Zine p. S81  abstract

Synthesis of Novel Azabenzimidazole Bridged bis-Coumarin Compounds, Investigation of Pancreatic Lipase Inhibitory Properties, and Docking Studies

Gülay Akyüz, Özlem Faiz, Mustafa Emirik, and Emre Menteşe p. S96  abstract

Synthesis, Structure, and In Vitro Pharmacological Evaluation of some New Pyrimidine-2-Sulfonamide Derivatives and Their Molecular Docking Studies on Human Estrogen Receptor Alpha and CDK2/Cyclin Proteins

Qassim A. H. Jaber, Ahmed Hassen Shentaif, Mohammed Almajidi, Iqrar Ahmad, Harun Patel, Abul Kalam Azad, Sulaiman Mohammed Alnasser, Hanan Ali Alatawi, Farid Menaa, Sulaiman Y.M. Alfaifi, Mohammed M. Rahman, Meser M. Ali, and S. J. Aditya Rao p. S106  abstract

Design, Synthesis, and Molecular Docking of a Novel Pyrimidine Terminal Alkyne Antitumor Agent

Tingting Fan, and Feng Jin p. S119  abstract

Novel Quinoxaline Derivatives: Design, Synthesis, Bioactive Evaluation, SARs, and Preliminary Antibacterial Mechanism

Zhongde Xie, Xuelian Dai, and Liqing Wang p. S132  abstract

Synthesis of 6-Alkylamino-2-alkylthio(alkoxy) Purine Derivatives: Antiplatelet Aggregation Activity Evaluation and 3D-QSAR Analysis

Shunlai Li, Pengyu Zheng, Yajing Ren, and Hongguang Du p. S146  abstract

Synthesis, Characterization, Antibacterial Evaluation, and Insecticidal Activity of Some Heterocyclic Compounds Containing Styrylpyridine Moiety

Y. A. El-Ossaily, E. A.-G. Bakhite, M. A. Gad, H. H. M. Abdu-Allah, S. Abuelhasan, O. F. Ibrahim, I. S. Marae, I. O. Althobaiti, N. M. M. Alanazi, N. S. Al-Muailkel, M. Y. El-Sayed, and M. M. Alanazi p. S159  abstract

Synthesis, Antitubercular, and Antifungal Activity of 2-(trifluoromethyl)-3-(substituted phenyl-1,3,4-oxadiazol-2-yl)-pyridine

B. K. Dhotre, S. V. Raut, M. Farooqui, S. B. Jadhav, and A. Pathan p. S171  abstract

COX-2 Enzyme Inhibitors Study and Efficacy Pharmacokinetic by Molecular Docking for some New Heterocyclic Rings Driver from Levofloxacin Drug

Muna Ismael Khalaf p. S179  abstract

Bovine Serum Albumin (BSA) Mediated Efficient One Pot Synthesis of 3,3′-(Phenylmethanediyl)bis(4-hydroxy-6-methyl-2H-pyran-2-one) Derivatives and Their Biological Studies

B. Manjunatha, Yadav D. Bodke, R. Kenchappa, P. Meghana, and P. V. Navaneethgowda p. S187  abstract

Design, 2D Qsar Studies, Molecular Docking, and Synthesis of Novel Triazole Derivatives intended as an Antifungal Agents

K. Yuvarani, N. Ramalakshmi, and S. Arunkumar p. S202  abstract

Replicative Senescence in Human Embryo Bone Marrow MSCs is Characterized by Changes in Cell Motility and Subcellular Localization of Rac1 and RhoA GTPases

A. V. Lukacheva, A. I. Gorb, A. S. Musorina, D. V. Kriger, G. G. Poljanskaya, and D. E. Bobkov p. S224  abstract

Huntington’s Disease Alters the Dermal Fibroblasts Secretome

M. Khotin, N. Kraskovskaya, P. Parfionova, N. Yudintceva, Y. Kolesnichenko, E. Ovcharenko, E. Repkin, S. Shabelnikov, A. Mittenberg, and N. Mikhailova p. S241  abstract