Contents

Russian Journal of Bioorganic Chemistry


Vol. 50, No. 5, 2024


Synthesis and Evaluation of Some Novel 1,3-Dimethylbarbituric Acid Derivatives as Potent Anti-Urease Agents: Comprehension through In Vitro, Molecular Docking, and DFT Investigations

Misbah Gul, Faheem Jan, Aftab Alam, Imtiaz Ahmad, Uzma Habib, Momin Khan, Abdullah F. AlAsmari, Fawaz Alasmari, Ajmal Khan, and Ahmed Al-Harrasi p. 1609  abstract

Exploring bis-Schiff Bases with Thiobarbiturate Scaffold: In Vitro Urease Inhibition, Antioxidant Properties, and In Silico Studies

Saba Gul, Safia Maab, Huma Rafiq, Aftab Alam, Munir Ur Rehman, Mohammad Assad, Abdullah F. AlAsmari, Fawaz Alasmari, Muhammad Ibrahim, and Momin Khan p. 1627  abstract

Discovering the DPPH Free Radical Scavenging Activity of Azine Derivatives Bearing Ethyl Phenyl Ketone Moiety

Munir Ur Rehman, Aftab Alam, Syed Adnan Ali Shah, Abid Ali, Qaisar Ali, Abdullah F. AlAsmari, Fawaz Alasmari, and Momin Khan p. 1639  abstract

Synthesis of Thioacetamide-Thiazoles as Anticholinesterase and Antioxidant Agents against Alzheimer’s Disease

Arti Soni, Ashwani Kumar, and Vivek Kumar p. 1646  abstract

Design, Synthesis, and Biological Evaluation of Novel Apigenin Derivatives as Potential Antitumor Agents

Bei-Qiao He, Xiao-Xiao Fan, Tian-Yu Zheng, Ya-Ting Gao, Xu Chen, Yong-Gang Liu, and Yuan-Yuan Zhang p. 1659  abstract

Synthesis and Importance of Coumarin Derivatives in Medicinal Chemistry: A Comprehensive Review

Mahima Samanth, and Mahesh Bhat p. 1672  abstract

ATP-Dependent LonBA Proteases of Bacilli and Clostridia

A. G. Andrianova, A. M. Kudzhaev, I. V. Smirnov, and T. V. Rotanova p. 1692  abstract

Boc/Bzl Solid-Phase Synthesis of Deltorphin II and Its Analogs without the Utilization of Anhydrous Hydrogen Fluoride

V. N. Azev, L. G. Mustaeva, E. Yu. Gorbunova, L. K. Baidakova, A. N. Chulin, L. N. Maslov, A. V. Mukhomedzyanov, М. В. Molchanov, and A. I. Miroshnikov p. 1701  abstract

Synthesis, Antimicrobial Evaluation, and Computational Study of Novel Fluorinated Benzofuran Derivatives

S. G. Dengale, K. K. Deshmukh, H. N. Akolkar, N. R. Darekar, M. H. Shaikh, V. M. Khedkar, and S. D. Kasar p. 1710  abstract

In Vitro Antibreast Cancer and Anti-EGFR Studies of Some Novel Benzimidazole-Piperazine Containing 1,2,3-Triazoles

Prasad Pinnoju, Sadanandam Kudikala, Manasa Scandakashi, Madavi Ramesh, and Sarasija Madderla p. 1724  abstract

Synthesis, Computational, and Photophysical Probing Studies on Mono-Azo Sulfonamides, and Their Antibacterial Activity

Pampapathi Shekharagouda, G. P. Mamatha, K. M. Pallavi, G. Nagaraju, Chethan Krishnamurthy, Vinodkumar P. Sajjan, M. S. Sushma, and Lohith Naik p. 1735  abstract

Advances in Drug Delivery Systems for Lipophilic Drug Paclitaxel: Developments, Challenges, and Opportunities (A Review)

Sumit Kumar, Aditi Arora, Vaishali Pant, Shramana Guchhait, Rajesh Kumar, Divya Mathur, and Brajendra K. Singh p. 1752  abstract

Synthesis and Characterization of Some New 2,3-Disubstituted Quinazolin-4(3H)-one Compounds, Investigation of Urease, and AChE Inhibition Properties, Molecular, and Docking Study

N. Ünal Karaali, G. Akyüz, and M. Emirik p. 1783  abstract

Truncated Hemolysin II and Cytotoxin K2 Forms of Bacillus cereus

A. S. Nagel, O. S. Vetrova, N. V. Rudenko, A. K. Surin, A. P. Karatovskaya, A. V. Zamyatina, N. A. Egorova, A. V. Siunov, Zh. I. Andreeva-Kovalevskaya, F. A. Brovko, and A. S. Solonin p. 1800  abstract

An Approach to the Synthesis of Cyclic Photocleavable RNA for Photoactivatable CRISPR/Cas9 System

E. V. Ivanskaya, M. I. Meschaninova, M. A. Vorobyeva, D. O. Zharkov, and D. S. Novopashina p. 1807  abstract

Synthesis, Antitubercular Evaluation of New 2,3-(4-Aminobenzamido)benzoic Acid Derivatives

Prashik B. Dudhe, Sujata P. Dudhe, Muthu K. Kathiravan, and Hardik G. Bhatt p. 1822  abstract

Synthesis of Some Novel (E)-1,5-Dimethyl-2-phenyl-4-(((2-arylimidazo[1,2-a]pyridin-3-yl)-methylene)amino)-1,2-dihydro-3H-pyrazol-3-one Derivatives: Exploring Their Antimicrobial Activity

Nilesh Kanzariya, Meet Sherashiya, Parth Barbhaya, Chandankumar Pashavan, and Yogesh Naliapara p. 1838  abstract

Design, Synthesis, and Anticancer Activities of Bakuchiol-1,3,5-triazine Derivatives

Rui Li, Ya-Min Ding, Tian Qin, Xuan-Yi Xue, Wei-Wei Liu, Rong-Bin Wei, Yuan-Fen Zhai, Gang Ding, and Da-Hua Shi p. 1851  abstract

Antidiabetic, Antidepressant, Antiparkinson’s, Neuroprotective, and Antioxidant Potentials of Novel Schiff Base Derivatives of a Lichen Metabolite, Usnic Acid

L. Yabo-Dambagi, A. Cakir, and A. Karaküçük-İyidoğan p. 1863  abstract

Design and Synthesis of Linear Acetamides as Cholesterol Lowering Agents

M. Sangeetha, Aathi Muthusankar, and J. Anitha p. 1882  abstract

Application of Time-Resolved Fluorescence Microscopy for Enhancing the Selectivity of Fluorogenic Dyes of the Arylidene–Imidazolone Series toward the Endoplasmic Reticulum

A. R. Gilvanov, A. Yu. Smirnov, S. A. Krasnova, I. D. Solovyev, A. P. Savitsky, Yu. A. Bogdanova, and M. S. Baranov p. 1896  abstract

Synthesis of SARS-CoV-2 Spike Glycoprotein Peptide Fragments and Study of Their Binding to Human Blood Cells

О. V. Gribovskaya, V. V. Yanchenko, A. M. Tsygankov, and V. P. Martinovich p. 1904  abstract

Structural and Functional Features of Protein–Polysaccharide Complexes Based on Cysteine Proteases and Hydrophilically Modified Chitosan

M. S. Lavlinskaya, A. V. Sorokin, S. S. Goncharova, M. G. Holyavka, M. S. Kondratyev, and V. G. Artyukhov p. 1917  abstract

Exploring the DPPH Radical Scavenging Potential in 5-Arylidene-N,N-diethylthiobarbiturates

Momin Khan, Munir Ur Rehman, Aftab Alam, Muhammad Ashraf, Uzma Salar, Khalid Mohammed Khan, Abdullah F. AlAsmari, and Fawaz Alasmari p. 1928  abstract

L-Proline Catalyzed Synthesis of Dihydropyrano[2,3-c]pyrazoles and Their Anti-Inflammatory Activity

K. J. Pansuriya, I. J. Modasiya, and G. G. Dubal p. 1935  abstract

Microwave-Assisted Synthesis of Pyridine-Conjugated 2-Methyl-6-(4-nitrophenyl)nicotine Hydrazide Schiff Base: Biological Screening of In Vitro Antimicrobial and In Silico ADMET Investigation

Parth Unjiya, Umang Patel, Hemal Parmar, Vaishali Rathod, Chandankumar Pashavan, and Manish Shah p. 1943  abstract

Development of the Contrasting Fluorescence Immunostaining Technique for 3D Imaging of Astrocyte Ultramorphology

K. E. Mochalov, O. I. Sutyagina, A. V. Altunina, D. O. Solovyeva, A. E. Efimov, V. A. Zhuchkov, S. P. Chumakov, and V. A. Oleinikov p. 1957  abstract

Features of the Amino Acid Composition of Gelatins from Organs and Tissues of Farm Animals (A Review)

S. Yu. Zaitsev p. 1966  abstract

3-Hydroxyquinazoline Derivatives, Analogues of Erastin, Induce Ferroptosis in Colorectal Cancer Cells

V. N. Osipov, A. A. Vartanyan, D. A. Khochenkov, D. V. Gusev, O. V. Fateenkova, D. S. Khachatryan, and L. M. Borisova p. 1980  abstract

SiO2 Nanoparticles Alter Basal Intracellular Calcium Concentration by Reducing TRPC1 Channel Expression in Human Retinal Pigment Epithelium Cell Line

A. H. Kaynar, F. Söğüt, Ş. N. Yılmaz, S. Yıldırımcan, and Ü. Çömelekoğlu p. 1991  abstract

Synthesis, In Vitro and In Silico Investigations of 4-(1H-Indol-3-yl)-N′-[(E/Z)-(phenyl-substituted)methylidene] as Effective Inhibitors of α-Glucosidase

M. Nazir, U. Khan, and M. Jahangir p. 1998  abstract

Synthesis, In Vitro and In Silico Evaluation of 3-(4, 5-Diphenyl-4H-1,2,4-triazol-3-yl)pyridine Derivatives As Potential Antimicrobial Agents

R. Dinkar, M. Yadav, A. Jain, N. Kumar, S. N. Mali, S. Kumar, B. Mathew, and S. Sharma p. 2013  abstract

Recent Progress of Sulfonamide-Indole/Carbazole Hybrids with the Anticancer Potential (A Review)

Ye Wang, Chaoyin Liu, and Zhi Xu p. 2024  abstract

Immobilization of Protein Probes on Biochips with Brush Polymer Cells

G. F. Shtylev, I. Yu. Shishkin, V. E. Shershov, V. E. Kuznetsova, D. A. Kachulyak, V. I. Butvilovskaya, A. I. Levashova, V. A. Vasiliskov, O. A. Zasedateleva, and A. V. Chudinov p. 2036  abstract

Generation of Active Amino Groups on the Surface of a Polyethylene Terephthalate Film and Their Quantitative Evaluation

G. F. Shtylev, I. Yu. Shishkin, S. A. Lapa, V. E. Shershov, V. E. Barsky, S. A. Polyakov, V. A. Vasiliskov, O. A. Zasedateleva, V. E. Kuznetsova, and A. V. Chudinov p. 2050  abstract

Detection of the IDH1/2 Gene Mutations in Tumor Samples with Low-Abundance Mutant Allele

V. O. Varachev, D. A. Guskov, O. Yu. Susova, A. P. Shekhtman, D. V. Rogozhin, S. A. Surzhikov, A. V. Chudinov, A. S. Zasedatelev, and T. V. Nasedkina p. 2058  abstract

Synthesis and Study Anti-Inflammatory Activity of Nicotinic Acid Hydrazones

О. А. Nurkenov, S. D. Fazylov, E. М. Satbayeva, Т. М. Seilkhanov, А. Zh. Mendibayeva, S. K. Kabiyeva, and Sh. N. Tursymbek p. 2066  abstract

Synthesis of Novel Dioxathiole-6,7-coumarin Hybrids As Cytosafe-Multifunctional Applicants: An In VitroIn Silico Study

Nameer Mazin Zeki, and Yasser Fakri Mustafa p. 2076  abstract

Erratum

Erratum to: Synthesis, Study Antimicrobial, and Antioxidant Agents of New Tetrazole Derivatives Containing 2-Amino-5-(4-nitrophenyl)-1,3,4-thiadiazol

Khadija Najah Zaidane, and Ahmed Wahed Naser p. 2092  abstract

Erratum to: Histopathological, Antioxidant, and Enzyme Activity of Boronic Incorporated Catechin Compound: Screening of Bioactivity with Molecular Docking Studies

Salih Paşa, Metin Atlan, Hamdi Temel, Burçin Türkmenoğlu, Abdulselam Ertaş, Aslı Okan, Seher Yilmaz, and Şükrü Ateş p. 2093  abstract