Contents

Russian Journal of Bioorganic Chemistry


Vol. 50, No. 2, 2024


Neurodegenerative Diseases: from the First CNS Drugs to New Treatments in Discovery (A Review)

Jean-Louis Kraus p. 273  abstract

Synthesis of Some New Coumarin-thiazolidine-2,4-dione-1,2,3-triazole Hybrids as Tubulin Targeting Anti-Lung Cancer Agents

B. Ramakrishna, B. Karthik, B. Ashok Kumar, and T. Kranthi Kumar p. 282  abstract

Synthesis of Morpholine Linked Indole-1,2,3-triazole Hybrids as In Vitro Tubulin Polymerization Inhibiting Agents

Prasad Pinnoju, Sadanandam Kudikala, Manasa Scandakashi, Madavi Ramesh, and Sarasija Madderla p. 293  abstract

Synthesis and Antimicrobial Activity of New Dihydropyrazolo[1,5-a]pyrimidine Derivatives

K. A. Joshi, H. B. Pandya, A. K. Mahida, I. J. Modasiya, and G. G. Dubal p. 304  abstract

Synthesis and Antitumor Activity Study of Novel Formononetin Derivatives

Zeping Luo, Liwei Pan, Xiuju Yin, and Hailin Chen p. 313  abstract

Synthesis and Evaluation of Antibacterial Properties of 1,2,3-Triazole Sulfonamide Derivatives

J. Y. Kong, X. Zhang, and G. S. Xuan p. 328  abstract

Synthesis, Characterization of Novel Thiazole Hydrazine Derivatives, and Inhibitory Action Against the VEGFR-2

V. A. Gore, D. N. Pansare, A. P. Sarkate, S. V. Tiwari, R. N. Shelke, S. V. Bhandari, and D. S. Bhagat p. 345  abstract

Antimicrobial Metabolites from Pig Nasal Microbiota

A. A. Baranova, Y. V. Zakalyukina, A. P. Tyurin, V. A. Korshun, O. A. Belozerova, M. V. Biryukov, A. V. Moiseenko, S. S. Terekhov, and V. A. Alferova p. 354  abstract

Diaryl Pyrazoline, 1,3,4-Oxadizole, and 1,2,4-Triazole Pharmacophore Hybridization: Design, Synthesis, HDAC Inhibition, and Caspase 3/7 Activation Studies

Abdullah Yahya Abdullah Alzahrani, Pratibha Gupta, Vijay Patil, Franz-Josef Meyer-Almes, D. V. Sokolova, V. S. Pokrovsky, and C. S. Ramaa p. 375  abstract

Investigation of the Effect of Tamoxifen on hERG1 Potassium Channel Gene Expression in MCF-7 Cell Line

P. Eroglu, F. Sogut, D. Yetkin, S. Yalin, U. Comelekoglu, S. N. Yilmaz, and S. Erdoğan p. 392  abstract

Proteinase Resistance of Carnosine, Pyrrolylcarnosine and Salicylcarnosine

K. V. Shevchenko, I. Yu. Nagaev, O. I. Kulikova, S. L. Stvolinsky, V. P. Shevchenko, and N. F. Myasoedov p. 401  abstract

Biocompatible Zinc Nanoparticles Synthesis from Ficus subincisa for a Sustainable Tomorrow: Characterization and Therapeutic Applications

Priyanka Pokhriyal, Amanpreet Kaur, Abha Shukla, Soniya Dhiman, and Himanshu Gupta p. 408  abstract

9-Chloro-5,9-dienoic and Other Fatty Acids from Marine Sponge Penares sp.

Е. А. Santalova, and S. А. Kolesnikova p. 418  abstract

Anti-Inflamatory Activities of Novel Chalcone Derivatives

Ergin Yalçın, Sedat Sevin, Recep Uyar, and Furkan Ayaz p. 432  abstract

Design, Synthesis, Computational, and In Vitro Cytotoxic Potential of Novel 5,7,8,9-Tetrahydrotetrazolo[5,1-b]quinazolines Analogs

Asief Mohammed, Shiva Kumar Gubbiyappa, and Rajasekhar Reddy Alavala p. 444  abstract

E. Coli Nissle 1917 Based Carrier for DNA Delivery into Colorectal Carcinoma Cells

N. Deeb, G. D. Otinov, A. Mohamed, E. R. Gandalipov, E. A. Kovtunov, and E. I. Koshel p. 459  abstract

Nanoparticles Based on Polyferulic and Polygentisic Acids as New Carriers of Anticancer Drugs

I. V. Smirnov, A. V. Lisov, A. N. Zvonarev, N. E. Suzina, A. S. Kazakov, and M. Y. Zemskova p. 467  abstract

Synthesis, Biological Evaluation, Molecular Docking, and Molecular Dynamic Simulation Studies of Some New 5-(3,4,5-Trimethoxybenzyl)pyrimidine-2,4-diamine (Trimethoprim) Derivatives via Modified Mannich-Type Reaction

Pavithra, Itte Pushpavathi, Kuntewale Mohiyouddin Mussuvir Pasha, and T. H. Maruthi Nayaka p. 485  abstract

Hybrid Antimicrobial Coating Based on Conjugate of Hyaluronic Acid with LL-37 Peptide for PEO-Modified Titanium Implants

L. V. Parfenova, Z. R. Galimshina, G. U. Gil’fanova, E. I. Alibaeva, T. M. Pashkova, O. L. Kartashova, R. G. Farrakhov, V. R. Aubakirova, and E. V. Parfenov p. 500  abstract

Borneol Induced Hepatotoxicity via Caspase-3 and Oxidative Stress Pathwaysin in Zebrafish

Xinjun Liao, Kun Jia, Lirong Huang, Zigang Cao, and Huiqiang Lu p. 508  abstract

Research and Optimization of the Synthesis of GdF3:Tb X-Ray Phosphors for X-Ray Photodynamic Therapy

P. Sh. Ustabaev, P. D. Zykova, V. V. Bakhmetev, and E. I. Leonova p. 522  abstract

Design, Synthesis, and Anti-Tumor Activity Evaluation In Vitro of 4,6,7–Trisubstituted Quinazoline Derivatives Containing Acrylamide Group

Gu Dongling, Yang Zichen, Wang Shihao, Chi Lingling, Yu Fuqiang, Wang Hao, Si Xiaojie, Gao Chao, Ke Yu, Liu Hongmin, and Zhang Qiurong p. 530  abstract

Finger-Actuated Microfluidic Platform for Colorimetric Isothermal Diagnostics of Neisseria meningitidis and Herpes Simplex Virus

L. A. Shkodenko, V. O. Laushkina, M. S. Rubel, and E. Sergeeva p. 544  abstract

Synthesis and Hypoglycemic Activity of New Nicotinonitrile-Furan Molecular Hybrids

D. A. Tilchenko, E. Yu. Bibik, V. V. Dotsenko, S. G. Krivokolysko, K. A. Frolov, N. A. Aksenov, and I. V. Aksenova p. 554  abstract

Synthesis and Biological Evaluation of 2-(6-Phenylimidazo[2,1-b][1,3,4]thiadiazol-2-yl)benzo[d]thiazole Derivatives as EGFR Targeting Anticancer Agents

Boda Mahipal Reddy, Midde Sridhar, Mekala Himabindu, K. Bhaskar, G. V. R. Sai Madhukar, T. Karunakar, Sudhakar Reddy Baddam, and Mamatha Kasula p. 571  abstract

Composition and Pathogenic Potential of Mucosal Microbiota in Ulcerative Colitis

S. A. Tsvetikova, E. E. Kruglov, L. G. Danilov, D. S. Zilov, Yu. V. Myakisheva, M. A. Makarova, L. A. Kaftyreva, and E. I. Koshel p. 582  abstract

Stimulatory Effect on Mice by Bacterial Exopolysaccharide, Colanic Acid

S. A. Tsvetikova, A. A. Zabavkina, V. G. Nikonorova, S. A. Tsymbal, M. S. Dukhinova, V. V. Chrishtop, and E. I. Koshel p. 594  abstract

Design, Synthesis, and Biological Evaluation of a New Series of 2,4-Position Modified Pyrimidine Derivatives

L. Chen, Z. D. Yao, Y. Chen, and L. Zhao p. 604  abstract

Arylidene-Imidazolones and Their Acyclic Analogue as Fluorescent Sensors of Metal Ions

S. A. Krasnova, E. R. Zaitseva, D. I. Rudik, D. S. Ivanov, A. A. Mikhaylov, and M. S. Baranov p. 617  abstract

Erratum

Erratum to: A New Approach to the Synthesis of Anti-Reverse Cap Analog (ARCA) 2mGpppG

A. L. Kayushin, K. V. Antonov, E. V. Dorofeeva, M. Ya. Berzina, A. O. Arnautova, I. A. Prohorenko, A. I. Miroshnikov, and I. D. Konstantinova p. 625  abstract

Erratum to: Pyrazinamide Analogs Designed for Rational Drug Designing Strategies Against Resistant Tuberculosis (A Review)

Xinyu Wang, Hongshang Hu, Wenhao Zhou, Jingxian Gongye, Ting Wang, and Juan Xu p. 626  abstract