Contents

Russian Journal of Bioorganic Chemistry

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Vol. 50, No. 1, 2024

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A New Approach to the Synthesis of Anti-Reverse Cap Analog (ARCA) ^2mGpppG

A. L. Kayushin, K. V. Antonov, E. V. Dorofeeva, M. Ya. Berzina, A. O. Arnautova, I. A. Prohorenko, A. I. Miroshnikov, and I. D. Konstantinova p. 1  abstract

Pyrazinamide Analogs Designed for Rational Drug Designing Strategies Against Resistant Tuberculosis (A Review)

Xinyu Wang, Hongshang Hu, Wenhao Zhou, Jingxian Gongye, Ting Wang, and Juan Xu p. 8  abstract

Synthesis, Characterization, and Study of Anticancer Activities of New Schiff Bases and 1,3-Oxazepine Containing Drug

Rana Abid Ali, Luma S. Ahamed, and Shaima Ibraheem Chyad AL-Khazraji p. 28  abstract

Synthesis of Novel 2-((3-(Benzofuran-2-yl)-1-phenyl-1H-pyrazol-4-yl)methylene)hydrazinyl-4-phenylthiazole: Potent EGFR Targeting Anticancer Agents

Sateesh Amudala, Rambabu Palabindela, Srinu Bhoomandla, N Kotilingaiah, Jonnala Sandhya, and Jyothi Mandala p. 34  abstract

Surfactants as a Means of Delivering a Reporter Genetic Construct Based on Binase Suicide Gene to Tumor Cells

E. V. Dudkina, E. A. Vasilieva, V. V. Ulyanova, L. Ya. Zakharova, and O. N. Ilinskaya p. 45  abstract

Participation of the Transcription Factor CREB1 in the Regulation of the Mdh2 Gene Encoding Malate Dehydrogenase in the Liver of Rats with Alloxan-Induced Diabetes

A. T. Eprintsev, K. R. Romanenko, and N. V. Selivanova p. 56  abstract

Assessing the Potential of Vitamin Drug Conjugate for Its Activity against Infectious Disease

R. P. Bhole, P. C. Bhondave, and R. V. Chikhale p. 64  abstract

Synthesis of Novel N-Acylhydrazones Derived from 3,5-Dinitrobenzohydrazide and Evaluation of Their Anticholinesterase and Antioxidant Activities

Reşit Çakmak, Ercan Çınar, Eyüp Başaran, Gülsüm Tuneğ, Sevcan İzgi, and Mehmet Boğa p. 76  abstract

Synthesis, Characterization of Formazan Derivatives from Isoniazid and Study Their Antioxidant Activity and Molecular Docking

W. K. Damdoom, and O. H. R. Al-Jeilawi p. 86  abstract

Isolation, Physico-Chemical Characteristics, and Acute Toxicity Evaluation of Water-Soluble Polysaccharide from Basidial Raw Material Ganoderma lucidum

S. B. Khaytmetova, A. S. Turaev, G. A. Khalilova, and B. I. Muhitdinov p. 95  abstract

Tetrahedral Boronate Ester as Regulators of Inflammation and Adhesion in ox-LDL Induced Atherosclerotic Model

U. Degirmenci, A. Kilic, R. Söylemez, and M. Yildirim p. 106  abstract

Synthesis of Steroid Tracers by an Oxime Ligation Method and Their Use in Fluorescent Polarisation Immunoassay

I. A. Prokhorenko, D. A. Glushchenko, E. L. Gulyak, I. V. Mikhura, V. A. Korshun, L. I. Mukhametova, and S. A. Eremin p. 116  abstract

Benzothiophene Schiff Bases Disrupt Cytoplasmic Membrane Integrity of Gram-Positive and -Negative Bacteria Cells

Bengü Ergüden, Hatice Büşra Lüleci, and Yasemin Ünver p. 128  abstract

Synthesis, Spectral Identification of Some New Schiff Bases, and Evaluation of Their Antibacterial Activity and Inhibitory Effect on Proinflammatory Cytokines (IL-1β, TNF), and DNA Ligase

Israa A. Alhasan Hamdan, Alaa Abd Alhasan Hamdan, and Rasha A. Abidalmutalib Aljabawi p. 138  abstract

Synthesis and Anti-Mycobacterium Activity of Some New N-Rich Heterocyclic Derivatives and Their Molecular Docking, and DFT Studies

Raghavendra Hegde, Itte Pushpavathi, Talavara Venkatesh, O. Nagaraja, and S. Ravi Kumar p. 147  abstract

Design and Synthesis of Benzo-Spirocyclic Derivatives as Potent PARP-1 Inhibitors

Shu Jia, Ling Yu, Jing-yi Zhao, Shuai Li, and Xin He p. 162  abstract

Synthesis, Identification, Antioxidant, Molecular Docking, and In Silico ADME Study for Some New Derivatives Containing Thiourea Moiety

Asmaa Abdulbaqi Maryoosh, and Oday H. R. Al-Jeilawi p. 170  abstract

Synthesis of Chromeno[2,3-d]pyrimidine-2,4(3H)-dion Derivatives Fused with Indole Moiety as Potent Biological Agents

P. V. Navaneethgowda, Y. D. Bodke, B. Manjunatha, N. D. Satyanarayan, and N. B. Nippu p. 181  abstract

Synthesis and Biological Evaluation of Coumarin-Amino Acid-Benzotriazole Conjugates

Emre Menteşe, Nedime Çalışkan, Bahar Bilgin Sökmen, and Gülay Akyüz p. 191  abstract

New Coumarin-Metronidazole Composites: Synthesis, Biocompatibility, and Anti-anaerobic Bacterial Activity

Yasser Fakri Mustafa p. 201  abstract

Acetylcholine Inhibitory Study of Novel Thio Linked Coumarin-Benzimidazole Derivatives: Design, Synthesis, Computational, and In Silico Molecular Docking Studies

T. H. Maruthi Nayaka, Itte Pushpavathi, Pavithra, and Y. R. Nagesh p. 211  abstract

Novel Bipyrazole Targeting Dual CDK-2 and VEGFR-2 Kinases: Synthesis, Anticancer Evaluation, and In Silico Studies

E. S. Nossier, N. M. Khalifa, H. H. Fahmy, M. M. F. Ismail, H. M. El-Sahrawy, and M. M. Ali p. 227  abstract

Effective Microwave-Assisted Synthesis of 2-Chloro-5,6-dimethyl-3-(((substituted-benzylidene)hydrazono)methyl)-quinoline and Its Biological Assessment

N. K. Vegal, T. D. Bhatt, K. Kachhot, and H. S. Joshi p. 239  abstract

2,5-Dimethoxy-Benzylidene-Rhodanine and Its Acyclic Analogues as Selective Fluorogenic Dyes for Lipid Droplets of Living Cells

S. A. Krasnova, Yu. A. Bogdanova, A. I. Sokolov, I. N. Myasnyanko, A. Yu. Smirnov, and M. S. Baranov p. 251  abstract

Aminocoumaranones as Chemiluminescence Indicators of the Urease Activity and Hydrogen Peroxide

A. Yu. Smirnov, N. S. Baleeva, A. S. Mishin, Yu. A. Bogdanova, and M. S. Baranov p. 260  abstract

Aryliden-Imidazolones as Fluorogens of NanoLuc Protein

E. R. Zaitseva, Yu. A. Bogdanova, N. S. Baleeva, A. Yu. Smirnov, and M. S. Baranov p. 267  abstract

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