Contents

Russian Journal of Bioorganic Chemistry

Vol. 47, No. 1, 2021

Synthetic Analogs of Streptococcus pneumoniae Capsular Polysaccharides and Immunogenic Activities of Glycoconjugates

M. L. Gening, E A. Kurbatova and N. E. Nifantiev p. 1  abstract

Glycoconjugate Vaccines for Prevention of Haemophilus influenzae Type b Diseases

E. A. Khatuntseva and N. E. Nifantiev p. 26  abstract

Protecting Groups as a Factor of Stereocontrol in Glycosylation Reactions

A. I. Tokatly, D. Z. Vinnitskiy, N. E. Ustuzhanina and N. E. Nifantiev p. 53  abstract

Carbohydrate Systems in Targeted Drug Delivery: Expectation and Reality

E. S. Shchegravina, A. A. Sachkova, S. D. Usova, A. V. Nyuchev, Yu. A. Gracheva and A. Yu. Fedorov p. 71  abstract

Selective Acetylation of the Primary Hydroxyl Group in Methyl D-Hexopyranosides with a Mixture of Acetic Anhydride and Acetic Acid

Y. E. Tsvetkov, D. V. Yashunsky and N. E. Nifantiev p. 99  abstract

Letter to the Editor

Chemical Examination of the Knotwood of Shorea robusta

D. E. Tsvetkov, A. S. Dmitrenok, Yu. E. Tsvetkov, R. Kumar, V. K. Varshney and N. E. Nifantiev p. 103  abstract

Anti-HIV and Antibacterial Activities of Novel 2-(3-Substituted-4-oxo-3,4-dihydroquinazolin-2-yl)-2,3-dihydrophthalazine-1,4-diones

M. T. Sulthana, K. Chitra, V. Alagarsamy, G. Saravanan and V. Raja Solomon p. 112  abstract

Antimycobacterial Activity, In Silico ADME Evaluation, and Docking Study of Novel Thiazolidinedione and Imidazolidinone Conjugates

V. T. Angelova, T. Pencheva, R. Buyukliev, E. K. Yovkova, I. Valkova, G. Momekov and V. Vulcheva p. 122  abstract

Heterocyclic Resveratrol Analogs. Synthesis and Physiological Activity: Part 1–Analogs Obtained by the Replacement of Aryl Residues with Heterocyclic Fragments

A. V. Semenov, E. V. Semenova and O. I. Balakireva p. 134  abstract

Design, Synthesis, and Anti-Breast Cancer Activity of Some Hybrid Molecules Containing Coumarin Moiety

Eman M. Radwan, Elsherbiny H. Elsayed, Mohamed Abd El-Moneim and Amal M. Youssef Moustafa p. 149  abstract

Synthesis, Molecular Docking, In Silico ADME Predictions, and Toxicity Studies of N-Substituted-5-(4-Chloroquinolin-2-yl)-1,3,4-Thiadiazol-2-Amine Derivatives as COVID-19 Inhibitors

Hanaa S. Mohamed, Walaa S. El-Serwy and Weam S. El-Serwy p. 158  abstract

Synthesis and Docking Studies of Novel Carbazole-Thiazolidinedione Hybrid Derivatives as Antibacterial Agents

L. Kamala, B. Sathish Kumar and P. V. Anantha Lakshmi p. 166  abstract

Synthesis, Design, and Biological Evaluation of Novel Diethylphenylcarbamothioylphosphonate

Ridha Ben Ali, Rania Omrani, Amal Ben Othman, Anis Raddaoui, Azaiez Ben Akacha and Michèle Véronique El May p. 174  abstract

Synthesis, Biological Evaluation, Molecular Docking, ADME Predictions and QSAR Studies of Novel 1,2-Diazet and Pyrrole Derivatives as Anti-Inflammatory Agents

Walaa S. El-Serwy, Weam S. El-Serwy, Neama A. Mohamed, Emad M. M. Kassem, Rasha E. Mostafa and Hanaa S. Mohamed p. 183  abstract

Synthesis, Molecular Docking, In Vitro Anti-Bacterial, and Anti-Cancer Activities of Some Novel Oxo-Spiro Chromene Schiff’s Bases

O. A. Lotlikar, S. N. Dandekar, M. M. V. Ramana and S. V. Rathod p. 199  abstract

New Diclofenac Derivatives as Anti-Microbial, Anti-Inflammatory Agents: Design, Synthesis, Biological Screening, and Molecular Docking Study

Mahmoud M. Hamed, Adel M. Kamal El-Dean, Shawkat A. Abdel-Mohsen and Mahmoud S. Tolba p. 208  abstract

Synthesis and Acaricidal Activity of Aryl-Spirobutyrolactone Derivatives against Spider Mites under Greenhouse and Field Conditions

L. K. Zhong, J. Yuan, X. H. Liu, T. M. Xu and C. X. Tan p. 221  abstract

Transformations of the Chromophore in the Course of Maturation of a Chromoprotein from Actinia equina

A. A. Pakhomov, A. A. Pastukhova, G. V. Tishkin and V. I. Martynov p. 230  abstract

Thermodynamic and Kinetic Parameters of Thermostable Alkaline Phosphatase from Geobacillus pallidus P26

S. Y. Çelik and H. Ilhan p. 236  abstract

Physicochemical Properties of Photoconvertible Fluorescent Protein from Montastraea cavernosa

A. Yu. Frolova, A. A. Pakhomov and V. I. Martynov p. 244  abstract

Transcriptome Profiles in the Spleen of the Chinese Giant Salamander (Andrias davidianus) Challenged with Citrobacter freundii

X. C. Gao, S. H. Niu, Y. Huang, J. L. Xiong and H. T. Ren p. 252  abstract

Inhibitory Evaluation and Molecular Docking Analysis of Benzenesulfonamides on Carbonic Anhydrase II

A. M. Zhang, N. Wei, X. F. Liu, M. G. Wu and G. S. Xuan p. 261  abstract

Influence of Subchronic Administration of the HLDF-6 Peptide on an Efficacy of the Exploratory Behavior of Inbred Mice of the Balb/c and C57Bl/6 Strains

G. I. Kovalev, E. V. Vasileva, R. M. Salimov, Yu. A. Zolotarev, A. K. Dadayan, A. P. Bogachouk and V. M. Lipkin p. 270  abstract

The Role of Linker Histones in Carcinogenesis

A. V. Lyubitelev, M. P. Kirpichnikov and V. M. Studitsky p. 278  abstract

Cytotoxic Activities and QSAR Studies of Diterpenoid Isosteviol Derivatives as Anti-Esophageal Agents

Cong-Jun Liu, Yu-Fei Wang, Jian-Hua Yao, Yan-Ping Liu, Qiao-Juan Jiang and Pan-Ping Liu p. 288  abstract

Gallocyanine as a Fluorogen for the Identification of NADPH-Dependent Production of Superoxide Anion Radical by Blood Cells

O. M. Panasenko, V. E. Reut, I. V. Borodina, D. S. Matyushkina, V. A. Ivanov, D. V. Grigorieva, I. V. Gorudko, A. V. Sokolov and S. N. Cherenkevich p. 299  abstract

Antitumor Activity of Monasnicotinic Acid Isolated from the Fungus Aspergillus cavernicola

G. K. Rystsov, T. V. Antipova, K. V. Zaitsev and M. Yu. Zemskova p. 307  abstract

3D-Pharmacophore Modeling, Molecular Docking, and Virtual Screening for Discovery of Novel CDK4/6 Selective Inhibitors

Amany Belal p. 317  abstract

Styrene Derivatives of Indole and Pyranone as Fluorogenic Substrates for FAST Protein

A. I. Sokolov, I. N. Myasnyanko, N. S. Baleeva and M. S. Baranov p. 334  abstract